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40건 · 전체 패밀리
- 화합물DM1 (mertansine)Maytansinoid
- 패밀리DM1 / maytansinoid payload familyMaytansinoid
- 화합물Gefitinib (Iressa)EGFR TKI
- 화합물Irinotecan (CPT-11)TOP1 inhibitor
- 패밀리MMAE (auristatin) payload familyADC payload
- 화합물MMAE (monomethyl auristatin E)ADC payload
- 화합물Osimertinib (Tagrisso)EGFR TKI
- 화합물Ribociclib (Kisqali)소분자
- 화합물SN-38 (active metabolite)TOP1 inhibitor
- 화합물SN-38 (irinotecan active)TOP1 inhibitor
- 화합물Sotorasib (Lumakras)KRAS inhibitor
- 화합물ALK macrocycle SAR analog소분자
- 화합물Auristatin E (parent)ADC payload
- 화합물BCR-ABL SAR methyl analog소분자
- 화합물BTK butynamide SAR analog소분자
- 화합물CDK amide-extended analog소분자
- 화합물CDK SAR piperazine analog소분자
- 화합물Daraxonrasib analog 03 (warhead methyl)KRAS inhibitor
- 화합물DM1 N-de methyl analogMaytansinoid
- 화합물DXd membrane-permeability SAR analogTOP1 inhibitor
- 화합물EGFR morpholine SAR analogEGFR TKI
- 화합물EGFR SAR analog (acrylamide branch)EGFR TKI
- 화합물KRAS chloro-bridge analogKRAS inhibitor
- 패밀리KRAS G12C inhibitor chemical landscapeKRAS inhibitor
- 화합물KRAS piperazine SAR analogKRAS inhibitor
- 화합물KRAS SAR analog A (F-aryl walk)KRAS inhibitor
- 화합물KRAS SAR analog B (from analog A)KRAS inhibitor
- 화합물MMAE C-terminal SAR analogADC payload
- 화합물MMAE-PEG4 analogADC payload
- 화합물Osimertinib active metabolite (AZ7550)EGFR TKI
- 화합물PARP fluoro-aryl analog소분자
- 화합물PARP SAR indole analog소분자
- 화합물Sacituzumab govitecan (Trodelvy)Maytansinoid
- 화합물SG3199 (PBD dimer warhead)ADC payload
- 화합물SMCCKRAS inhibitor
- 화합물SMCC-DM1 (linker-payload)Maytansinoid
- 패밀리SN-38 / irinotecan (TOP1) small-molecule seriesTOP1 inhibitor
- 화합물SN-38 ADC linker-payload designTOP1 inhibitor
- 화합물SN-38 lipophile analogTOP1 inhibitor
- 화합물SN-38 payload (cross-family)Maytansinoid
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