KRAS inhibitor
- ADC: 2
- Payload: 3
- Derivative: 5
- Drug: 1
- Scaffold: 1
- Linker: 3
Payload: daraxon-payload-p1, daraxon-payload-p2, daraxon-payload-p3
KRAS G12C covalent inhibitor core and derived small molecules, ADC payloads, linkers, and assembled ADCs.
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- Drug: 6
- Scaffold: 1
- Derivative: 5
- Payload: 1
Payload: kras-adc-payload-1
Shared acrylicamide / warhead chemotype from core scaffold to sotorasib, adagrasib, daraxonrasib and SAR analogs.
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- Drug: 4
- Derivative: 2
- Scaffold: 1
Non-covalent and RAS(ON) chemotypes targeting KRAS G12D — MRTX1133, RMC-6236, RMC-9805 and SAR analogs.
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