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Mechanism classes

Search often arrives by mechanism, not by a single INN. Each hub groups a class summary, representative drugs, and family/compound permalinks across the catalog.

  • KRAS G12C covalent inhibitorsKRAS G12C 공유결합 저해제3 families · 35 compounds
  • EGFR tyrosine kinase inhibitorsEGFR 타이로신키나제 저해제1 families · 11 compounds
  • ADC payloads (auristatin, exatecan, maytansinoid)ADC payload — MMAE · DXd · DM17 families · 58 compounds
  • PARP inhibitorsPARP 저해제1 families · 7 compounds
  • CDK4/6 inhibitorsCDK4/6 저해제1 families · 6 compounds
  • BTK inhibitorsBTK 저해제1 families · 6 compounds
  • ALK / ROS1 inhibitorsALK / ROS1 TKI1 families · 6 compounds
  • BRAF / MEK inhibitorsBRAF / MEK 저해제1 families · 7 compounds
  • BCR-ABL tyrosine kinase inhibitorsBCR-ABL TKI1 families · 7 compounds
  • RET / MET / NTRK inhibitorsRET / MET / NTRK TKI1 families · 8 compounds
  • PI3K / AKT / mTOR inhibitorsPI3K / AKT / mTOR1 families · 7 compounds
  • PROTAC degradersPROTAC / 분해제1 families · 7 compounds
  • JAK inhibitorsJAK 저해제1 families · 6 compounds
  • BCL-2 inhibitorsBCL-2 저해제1 families · 6 compounds
  • Taxanes / microtubule agents탁산 / 미세소관 제제1 families · 6 compounds
  • ADC linkersADC 링커1 families · 8 compounds
  • PCSK9 inhibitorsPCSK9 / LDL-C1 families · 9 compounds
  • GLP-1 / incretin agonistsGLP-1 / 인크레틴1 families · 10 compounds
  • SGLT2 inhibitorsSGLT2 저해제1 families · 6 compounds
  • Statins / HMG-CoA reductase스타틴 / HMG-CoA 환원효소1 families · 6 compounds
  • SSRI / SNRI antidepressantsSSRI / SNRI 항우울제1 families · 8 compounds
  • GABAergic anxiolytics불안 · GABA 벤조디아제핀1 families · 7 compounds
  • Antiepileptic drugs항경련제 (AED)1 families · 7 compounds
  • Cognitive / dementia agents인지 · 치매1 families · 6 compounds
  • Parkinson dopaminergic agents파킨슨 · 도파민 경로1 families · 11 compounds
  • ALS neuroprotectantsALS 신경보호1 families · 7 compounds
  • Gabapentinoids / neuropathic pain신경병증 · 가바펜티노이드1 families · 7 compounds
  • Atypical antipsychotics비정형 항정신병1 families · 6 compounds
  • Triptan antimigraine agents편두통 · 트립탄1 families · 7 compounds
  • CGRP receptor antagonists (gepants)편두통 · CGRP gepant1 families · 5 compounds
  • ADHD stimulants / non-stimulantsADHD 자극제·비자극제1 families · 8 compounds
  • Hypnotics / DORA수면 · hypnotic1 families · 8 compounds
  • S1P receptor modulators (MS)다발성 경화 · S1P 조절제1 families · 7 compounds
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