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KRAS G12C inhibitor chemical landscape

KRAS inhibitor

  • 화합물 13
  • 관계 58
  • SMILES 13/13
  • Drug: 6
  • Scaffold: 1
  • Derivative: 5
  • Payload: 1

Payload: kras-adc-payload-1

Shared acrylicamide / warhead chemotype from core scaffold to sotorasib, adagrasib, daraxonrasib and SAR analogs.

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