ADC payload
- Scaffold: 2
- ADC: 5
- Payload: 2
- Derivative: 2
- Linker: 1
Payload: mmae, mmaf
Microtubule-disrupting auristatin payloads derived from dolastatin 10 — widely used in approved and clinical ADCs.
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- Scaffold: 1
- Payload: 2
- Derivative: 1
- Linker: 1
- ADC: 1
Payload: duocarmycin-sa, seco-duocarmycin
Cyclopropapyrroloindole (CPI) DNA-alkylator payloads for ADCs — duocarmycin SA and seco forms.
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- Linker: 1
- Payload: 2
- Scaffold: 1
- ADC: 2
Payload: calicheamicin-gamma, nac-calicheamicin
Enediyne warhead for gemtuzumab ozogamicin (Mylotarg) and related ADCs.
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